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              PI-103

              Update:2014/12/6 20:08:40

                Item:PI-103
                Synonym:
                CAS No.:371935-74-9Special Grade:Biotech grade
                Formula:C19H16N4O3M.W.:348.36
              Order
                Product No.SizePriceBrand
                S1038-10mg10mg3650
                S1038-25mg25mg4689
                S1038-50mg50mg7530
                S1038-5mg5mg2520GBC
              Introduction
                PI-103有效抑制PI3K,可穿透細胞,是ATP競爭性抑制劑。PI-103作用于DNA-PK, p110α, mTORC1, PI3-KC2β, p110δ, mTORC2, p110β,和p110γ時,IC50分別為2, 8, 20, 26, 48, 83, 88, 150 nM。
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